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LCK protein kinase inhibitor A 770041, 5 mg  

LCK protein kinase inhibitor A 770041, 5 mg

N-(4-(1-(4-(4-acetylpiperazin-1-yl)cyclohexyl)-4-amino-1H-pyrazolo[3,4-d]pyrimidin-3-yl)-2-methoxyphenyl)-1-methyl-1H-indole-2-carboxamide

A 770041 is a selective and orally active Src-family Lck inhibitor

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PKI-A770041-005

Availability: within 3 days

202,50 €

Background: A 770041 is a selective and orally active Src-family Lck inhibitor; A-770041 is a 147 nM inhibitor of Lck (1 mM ATP) and is 300-fold selective against Fyn, the other Src family kinase involved in T-cell signaling.

Chemical formula: C34H39N9O3
Molecular weight: 621.73 g/mol
Purity: 99%
Appearance: White solid
Solubility: Soluble in DMSO
CAS Number: 869748-10-7

Manufacturer:  Axon Medchem BV

PLEASE NOTE: This product is designed for research purposes and can only be delivered to academic and business customers. 

References

H. Yamamoto et al. Bay K8644 differentiates between potential and receptor operated Ca2+ channels. Eur. J. Pharmacol. 1984, 102, 555-557.

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